Compile Data Set for Download or QSAR
Found 16 Enz. Inhib. hit(s) with all data for entry = 50027657
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50149871((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 10.2nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)copy SMILEScopy InChI
Affinity DataIC50: 11.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)copy SMILEScopy InChI
Affinity DataIC50: 11.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)copy SMILEScopy InChI
Affinity DataIC50: 20.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)copy SMILEScopy InChI
Affinity DataIC50: 21.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)copy SMILEScopy InChI
Affinity DataIC50: 29.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)copy SMILEScopy InChI
Affinity DataIC50: 87.7nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)copy SMILEScopy InChI
Affinity DataIC50: 94.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)copy SMILEScopy InChI
Affinity DataIC50: 226nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)copy SMILEScopy InChI
Affinity DataIC50: 278nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)copy SMILEScopy InChI
Affinity DataIC50: 542nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 574nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)copy SMILEScopy InChI
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed