Compile Data Set for Download or QSAR
Found 18 Enz. Inhib. hit(s) with all data for entry = 50029615
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286206((R)-5-tert-Butylcarbamoyl-4-(2-chloro-phenyl)-6-me...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286203(4-(2-Chloro-phenyl)-6-methyl-2-[2-(2-methyl-benzoi...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286211(4-(2-Chloro-phenyl)-6-methyl-2-[2-(2-methyl-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286206((R)-5-tert-Butylcarbamoyl-4-(2-chloro-phenyl)-6-me...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286204(4-(2-Chloro-phenyl)-6-methyl-2-[2-(2-methyl-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286207(4-(2-Chloro-phenyl)-6-methyl-2-[2-(2-methyl-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286201(4-(2-Chloro-phenyl)-6-methyl-5-(6-methyl-pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286212((R)-4-(2-Chloro-phenyl)-2-methyl-6-[2-(2,4,5-trime...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286209(4-(2-Chloro-phenyl)-6-methyl-5-phenylcarbamoyl-2-[...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286202((S)-4-(2-Chloro-phenyl)-2-methyl-6-[2-(2,4,5-trime...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286210(5-tert-Butylcarbamoyl-4-(2-chloro-phenyl)-6-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286205(4-(2-Chloro-phenyl)-6-methyl-2-[2-(2-methyl-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286208((S)-5-tert-Butylcarbamoyl-4-(2-chloro-phenyl)-6-me...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286202((S)-4-(2-Chloro-phenyl)-2-methyl-6-[2-(2,4,5-trime...)copy SMILEScopy InChI
Affinity DataIC50: 183nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286200(4-(2-Chloro-phenyl)-2-(4-imidazol-1-yl-phenyl)-6-m...)copy SMILEScopy InChI
Affinity DataIC50: 415nMAssay Description:Inhibitory effect on PAF induced platelets aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PMW