Compile Data Set for Download or QSAR
Found 16 Enz. Inhib. hit(s) with all data for entry = 50030240
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293023((Sar)WTLNSAGYLLGPKKKK | CHEMBL508036)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293024((Sar)WTLNSAGYLLGPKK(Lys-MPEG4)K | CHEMBL505299)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293030((Sar)WTLNSAGYLLGPKK(Lys-octanoyl)K | CHEMBL503900)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293029((Sar)WTLNSAGYLLGPKK(Lys-decanoyl)K | CHEMBL460706)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293028((Sar)WTLNSAGYLLGPKK(Lys-lauroyl)K | CHEMBL507733)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293027((Sar)WTLNSAGYLLGPKK(Lys-myristoyl)K | CHEMBL524678)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293026((Sar)WTLNSAGYLLGPKK(Lys-palmitoyl)K | CHEMBL507353)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293025((Sar)WTLNSAGYLLGPKK(Lys-stearoyl)K | CHEMBL450827)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293029((Sar)WTLNSAGYLLGPKK(Lys-decanoyl)K | CHEMBL460706)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293030((Sar)WTLNSAGYLLGPKK(Lys-octanoyl)K | CHEMBL503900)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293025((Sar)WTLNSAGYLLGPKK(Lys-stearoyl)K | CHEMBL450827)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293028((Sar)WTLNSAGYLLGPKK(Lys-lauroyl)K | CHEMBL507733)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293027((Sar)WTLNSAGYLLGPKK(Lys-myristoyl)K | CHEMBL524678)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293024((Sar)WTLNSAGYLLGPKK(Lys-MPEG4)K | CHEMBL505299)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293023((Sar)WTLNSAGYLLGPKKKK | CHEMBL508036)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293026((Sar)WTLNSAGYLLGPKK(Lys-palmitoyl)K | CHEMBL507353)copy SMILEScopy InChI
Affinity DataKi:  52nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3SD5PubMed