TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M4 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M4 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M5 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 6.00E+3nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 15 nM acetylcholine-induced calciu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 3.95E+5nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 15 nM acetylcholine-induced calciu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 10 uM acetylcholine-induced calciu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 715nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 10 uM acetylcholine-induced calciu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 10 uM acetylcholine-induced calciu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 15 nM acetylcholine-induced calciu...More data for this Ligand-Target Pair