Compile Data Set for Download or QSAR
Found 150 Enz. Inhib. hit(s) with all data for entry = 50034470
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362957(CHEMBL1946757)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362956(CHEMBL1946756)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362955(CHEMBL1946755)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362958(CHEMBL1946758)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362953(CHEMBL1947143)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362967(CHEMBL1947142)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362960(CHEMBL1946953)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362972(CHEMBL1946571)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362949(CHEMBL1947147)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362973(CHEMBL1946572)copy SMILEScopy InChI
Affinity DataIC50: 11.2nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362948(CHEMBL1947146)copy SMILEScopy InChI
Affinity DataIC50: 13.7nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362974(CHEMBL1946753)copy SMILEScopy InChI
Affinity DataIC50: 14.2nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362975(CHEMBL1946754)copy SMILEScopy InChI
Affinity DataIC50: 35.4nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362968(CHEMBL1947145)copy SMILEScopy InChI
Affinity DataIC50: 49.1nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362959(CHEMBL1946952)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362952(CHEMBL1946570)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362954(CHEMBL1947144)copy SMILEScopy InChI
Affinity DataIC50: 83.1nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362965(CHEMBL1947140)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362951(CHEMBL1946568)copy SMILEScopy InChI
Affinity DataIC50: 161nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362970(CHEMBL1946567)copy SMILEScopy InChI
Affinity DataIC50: 255nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362961(CHEMBL1946954)copy SMILEScopy InChI
Affinity DataIC50: 924nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362971(CHEMBL1946569)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+3nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362954(CHEMBL1947144)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362964(CHEMBL1947139)copy SMILEScopy InChI
Affinity DataIC50: 2.18E+3nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362962(CHEMBL1946955)copy SMILEScopy InChI
Affinity DataIC50: 3.66E+3nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362969(CHEMBL1946566)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362963(CHEMBL1947138)copy SMILEScopy InChI
Affinity DataIC50: 6.63E+3nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362966(CHEMBL1947141)copy SMILEScopy InChI
Affinity DataIC50: 6.94E+3nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362954(CHEMBL1947144)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C8More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362954(CHEMBL1947144)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362969(CHEMBL1946566)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362970(CHEMBL1946567)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362951(CHEMBL1946568)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362971(CHEMBL1946569)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362952(CHEMBL1946570)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362972(CHEMBL1946571)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362973(CHEMBL1946572)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362974(CHEMBL1946753)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362975(CHEMBL1946754)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362955(CHEMBL1946755)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362956(CHEMBL1946756)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362957(CHEMBL1946757)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362959(CHEMBL1946952)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362960(CHEMBL1946953)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362961(CHEMBL1946954)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362962(CHEMBL1946955)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362963(CHEMBL1947138)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362964(CHEMBL1947139)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362965(CHEMBL1947140)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362966(CHEMBL1947141)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human PPARalpha expressed in COS-1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P11PubMed
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