Affinity DataKi: 20nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 19.5+/-12.0More data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 117+/-46More data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 158+/-21More data for this Ligand-Target Pair
Affinity DataKi: 165nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membraneMore data for this Ligand-Target Pair
Affinity DataKi: 166nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 166+/-75More data for this Ligand-Target Pair
Affinity DataKi: 192nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membraneMore data for this Ligand-Target Pair
Affinity DataKi: 287nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 287+/-125More data for this Ligand-Target Pair
Affinity DataKi: 338nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 338+/-98More data for this Ligand-Target Pair
Affinity DataKi: 343nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 343+/-137More data for this Ligand-Target Pair
Affinity DataKi: 354nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 354+/-113More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 400+/-38More data for this Ligand-Target Pair
Affinity DataKi: 473nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 473+/-329More data for this Ligand-Target Pair
Affinity DataKi: 494nMAssay Description:Agonistic activity against adenosine A1 receptor in guinea pig isolated heartsMore data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 503+/-262More data for this Ligand-Target Pair
Affinity DataKi: 506nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 506+/-111More data for this Ligand-Target Pair
Affinity DataKi: 543nMAssay Description:Agonistic activity against adenosine A1 receptor in guinea pig isolated heartsMore data for this Ligand-Target Pair
Affinity DataKi: 604nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 604+/-241More data for this Ligand-Target Pair
Affinity DataKi: 614nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 614+/-78More data for this Ligand-Target Pair
Affinity DataKi: 894nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 894+/-659More data for this Ligand-Target Pair
Affinity DataKi: 913nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 913+/-517More data for this Ligand-Target Pair
Affinity DataKi: 1.14E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 1143+/-426More data for this Ligand-Target Pair
Affinity DataKi: 1.34E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 1571+/-245More data for this Ligand-Target Pair
Affinity DataKi: 1.67E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 1666+/-556More data for this Ligand-Target Pair
Affinity DataKi: 1.77E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 1773+/-209More data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 1945+/-1316More data for this Ligand-Target Pair
Affinity DataKi: 3.61E+3nMAssay Description:Agonistic activity against adenosine A1 receptor in guinea pig isolated heartsMore data for this Ligand-Target Pair
Affinity DataKi: 4.19E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CPX in guinea pig DDT membrane; 4191+/-922More data for this Ligand-Target Pair
Affinity DataKi: 4.39E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membraneMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 5497+/-180More data for this Ligand-Target Pair
Affinity DataKi: 5.86E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 5855+/-1208More data for this Ligand-Target Pair
Affinity DataKi: 6.25E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 6250+/-1767More data for this Ligand-Target Pair
Affinity DataKi: 7.29E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 7292+/-3241More data for this Ligand-Target Pair
Affinity DataEC50: 41nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 543+/-182More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 3612+/-1937More data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+3nMAssay Description:Agonistic activity against adenosine A1 receptor in guinea pig isolated heartsMore data for this Ligand-Target Pair