Affinity DataKi: 0.350nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]methylscopolamine [3H]NMS from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:The compound was evaluated for the inhibition human of Butyrylcholinesterase IMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:The compound was evaluated for the inhibition human of ButyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:The compound was evaluated for the inhibition human of ButyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of human acetylcholinesterase-IMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:The compound was evaluated for the inhibition human of ButyrylcholinesteraseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]pirenzepine binding to Muscarinic acetylcholine receptor M1 of mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:The compound was evaluated for the inhibition human of ButyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:The compound was evaluated for the inhibition human of Butyrylcholinesterase IMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:The compound was evaluated for the inhibition of human AcetylcholinesteraseMore data for this Ligand-Target Pair