Compile Data Set for Download or QSAR
Found 18 Enz. Inhib. hit(s) with all data for entry = 50036192
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043326(CHEMBL438733 | c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0930nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043322(CHEMBL427748 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)copy SMILEScopy InChI
Affinity DataIC50: 0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368776(CHEMBL1790962)copy SMILEScopy InChI
Affinity DataIC50: 0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368773(CHEMBL1790959)copy SMILEScopy InChI
Affinity DataIC50: 0.180nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368774(CHEMBL1790963)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368775(CHEMBL1790960)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368772(CHEMBL2373291)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368774(CHEMBL1790963)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368776(CHEMBL1790962)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368777(CHEMBL2373292)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043324(CHEMBL411171 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368777(CHEMBL2373292)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50368772(CHEMBL2373291)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043322(CHEMBL427748 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)copy SMILEScopy InChI
Affinity DataIC50: 0.75nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043326(CHEMBL438733 | c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-...)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043324(CHEMBL411171 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8MPCPubMed