Found 32 Enz. Inhib. hit(s) with all data for entry = 50037022 
Affinity DataKi: 0.0230nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.47nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.79nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 4.67nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.46nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 34.1nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 64.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 119nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 237nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 299nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 645nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 654nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 772nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.43E+3nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Bradykinin receptor B2-mediated contractions of rat uterus smooth muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Bradykinin receptor B2-mediated contractions of rat uterus smooth muscleMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonism of the [Ca2+] efflux actions of the human Bradykinin receptor B2 (SK-N-SH neuroblastoma)More data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonism of the [Ca2+] efflux actions of human Bradykinin receptor B2 (WI38 fibroblasts)More data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Antagonism of the [Ca2+] efflux actions of the human Bradykinin receptor B2 (WI38 fibroblasts)More data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences
Curated by ChEMBL
Novartis Institute for Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Antagonism of the [Ca2+] efflux actions of human Bradykinin receptor B2 (SK-N-SH neuroblastoma)More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibition of increase in [Ca2+] efflux from NG108-15 cells caused by activation of rat Bradykinin receptor B2More data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Inhibition of increase in [Ca2+] efflux from NG108-15 cells caused by activation of rat Bradykinin receptor B2More data for this Ligand-Target Pair
