TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human Cdc2 kinase PY15 phosphorylation in HT29 cells by Western blotMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human Cdc2 kinase PY15 phosphorylation in HT29 cells by Western blotMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human Cdc2 kinase PY15 phosphorylation in HT29 cells by Western blotMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2ZS2XC3PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2ZS2XC3PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human Wee1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human Cdc2 kinase PY15 phosphorylation in HT29 cells by Western blotMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
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