Compile Data Set for Download or QSAR
Found 32 Enz. Inhib. hit(s) with all data for entry = 50039509
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379214(CHEMBL2011291 | US9416123, 6)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379214(CHEMBL2011291 | US9416123, 6)copy SMILEScopy InChI
Affinity DataIC50: 113nMAssay Description:Inhibition of wild type EGFR using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379218(CHEMBL2011304)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379214(CHEMBL2011291 | US9416123, 6)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of wild type B-Raf using MEK1-KM as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379214(CHEMBL2011291 | US9416123, 6)copy SMILEScopy InChI
Affinity DataIC50: 399nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379227(CHEMBL2011293 | US9416123, 7)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379224(CHEMBL2011297 | US9416123, 11)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379225(CHEMBL2011295 | US9416123, 9)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379226(CHEMBL2011294 | US9416123, 8)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379218(CHEMBL2011304)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379228(CHEMBL2011292 | US9416123, 5)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379223(CHEMBL2011298 | US9416123, 12)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379216(CHEMBL2011296 | US9416123, 10)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379222(CHEMBL2011299 | US9416123, 14)copy SMILEScopy InChI
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379223(CHEMBL2011298 | US9416123, 12)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379217(CHEMBL2011305 | US9416123, 20)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379215(CHEMBL2011301 | US9416123, 18)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379227(CHEMBL2011293 | US9416123, 7)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379226(CHEMBL2011294 | US9416123, 8)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379217(CHEMBL2011305 | US9416123, 20)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379222(CHEMBL2011299 | US9416123, 14)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379220(CHEMBL2011302 | US9416123, 16)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379215(CHEMBL2011301 | US9416123, 18)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379228(CHEMBL2011292 | US9416123, 5)copy SMILEScopy InChI
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379216(CHEMBL2011296 | US9416123, 10)copy SMILEScopy InChI
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379220(CHEMBL2011302 | US9416123, 16)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379225(CHEMBL2011295 | US9416123, 9)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379219(CHEMBL2011303 | US9416123, 19)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379224(CHEMBL2011297 | US9416123, 11)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379221(CHEMBL2011300 | US9416123, 15)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379219(CHEMBL2011303 | US9416123, 19)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza

Curated by ChEMBL
LigandPNGBDBM50379221(CHEMBL2011300 | US9416123, 15)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8N18PubMed