Compile Data Set for Download or QSAR
Found 90 Enz. Inhib. hit(s) with all data for entry = 50039522
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379402(CHEMBL2012014)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379423(CHEMBL2012038)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379401(CHEMBL2011946)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379398(CHEMBL2011952)copy SMILEScopy InChI
Affinity DataKi:  320nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379396(CHEMBL2011950)copy SMILEScopy InChI
Affinity DataKi:  430nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379416(CHEMBL2012030)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379410(CHEMBL2012023)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379391(CHEMBL2012037)copy SMILEScopy InChI
Affinity DataKi:  900nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379425(CHEMBL2012040)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379415(CHEMBL2012029)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379418(CHEMBL2012032)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379413(CHEMBL2012027)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379414(CHEMBL2012028)copy SMILEScopy InChI
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379426(CHEMBL2012041)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379393(CHEMBL2011947)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379427(CHEMBL2012044)copy SMILEScopy InChI
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379405(CHEMBL2012017)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379393(CHEMBL2011947)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by manual whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379389(CHEMBL2010816)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379423(CHEMBL2012038)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379427(CHEMBL2012044)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379393(CHEMBL2011947)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by manual whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379413(CHEMBL2012027)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379426(CHEMBL2012041)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379425(CHEMBL2012040)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379396(CHEMBL2011950)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379427(CHEMBL2012044)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379425(CHEMBL2012040)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379396(CHEMBL2011950)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379428(CHEMBL2012039)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379415(CHEMBL2012029)copy SMILEScopy InChI
Affinity DataIC50: 590nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379405(CHEMBL2012017)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379405(CHEMBL2012017)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379414(CHEMBL2012028)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379389(CHEMBL2010816)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by manual whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379426(CHEMBL2012041)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379423(CHEMBL2012038)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379414(CHEMBL2012028)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379418(CHEMBL2012032)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379389(CHEMBL2010816)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379391(CHEMBL2012037)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379390(CHEMBL2012042)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379402(CHEMBL2012014)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379416(CHEMBL2012030)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379393(CHEMBL2011947)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human ERG by PatchXpress volatage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379389(CHEMBL2010816)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by manual whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379415(CHEMBL2012029)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379412(CHEMBL2012026)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379428(CHEMBL2012039)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.5 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379410(CHEMBL2012023)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at human partially inactivated NaV 1.7 channel expressed in HEK293 cells by PatchXpress voltage patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S183H3PubMed
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