Compile Data Set for Download or QSAR
Found 128 Enz. Inhib. hit(s) with all data for entry = 50039524
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379458(CHEMBL2012273)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379439(CHEMBL2012301)copy SMILEScopy InChI
Affinity DataKi:  320nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379455(CHEMBL2012269)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379438(CHEMBL2012300)copy SMILEScopy InChI
Affinity DataKi:  680nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379467(CHEMBL2012293)copy SMILEScopy InChI
Affinity DataKi:  730nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379452(CHEMBL2012266)copy SMILEScopy InChI
Affinity DataKi:  930nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379457(CHEMBL2012272)copy SMILEScopy InChI
Affinity DataKi:  950nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379465(CHEMBL2012291)copy SMILEScopy InChI
Affinity DataKi:  980nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379444(CHEMBL2012246)copy SMILEScopy InChI
Affinity DataKi:  990nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379437(CHEMBL2012299)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379469(CHEMBL2012295)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379471(CHEMBL2012260)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379470(CHEMBL2012277)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379450(CHEMBL2012263)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379440(CHEMBL2012179)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379448(CHEMBL2012259)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379442(CHEMBL2012181)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379436(CHEMBL2012298)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379466(CHEMBL2012292)copy SMILEScopy InChI
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379459(CHEMBL2012274)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379456(CHEMBL2012271)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379464(CHEMBL2012290)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379454(CHEMBL2012268)copy SMILEScopy InChI
Affinity DataKi:  2.46E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379441(CHEMBL2012180)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379431(CHEMBL2012178)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379453(CHEMBL2012267)copy SMILEScopy InChI
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379468(CHEMBL2012294)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379451(CHEMBL2012265)copy SMILEScopy InChI
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379437(CHEMBL2012299)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379448(CHEMBL2012259)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379457(CHEMBL2012272)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379456(CHEMBL2012271)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379448(CHEMBL2012259)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379436(CHEMBL2012298)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379438(CHEMBL2012300)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379441(CHEMBL2012180)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379458(CHEMBL2012273)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379459(CHEMBL2012274)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379466(CHEMBL2012292)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379451(CHEMBL2012265)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379436(CHEMBL2012298)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379437(CHEMBL2012299)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379458(CHEMBL2012273)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379442(CHEMBL2012181)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379440(CHEMBL2012179)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379457(CHEMBL2012272)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379449(CHEMBL2012262)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379440(CHEMBL2012179)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379441(CHEMBL2012180)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50379431(CHEMBL2012178)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Antagonist activity at 20% inactivated human NaV1.7 channel by electrophysiology-based screening assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM59GCPubMed
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