Compile Data Set for Download or QSAR
Found 127 Enz. Inhib. hit(s) with all data for entry = 50040289
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.240nMAssay Description:Inhibition of human recombinant JAK3 kinase domain using FITC-KGGEEEEYFELVKK as substrate by peptide mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391993(CHEMBL2152297)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition of JAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391996(CHEMBL2152300)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391993(CHEMBL2152297)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392011(CHEMBL2152401)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.680nMAssay Description:Inhibition of human recombinant GST-tagged JAK1 using 5-FAM-KKSRGDYMTMQIG as substrate by peptide mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391993(CHEMBL2152297)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of JAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.990nMAssay Description:Inhibition of human recombinant JAK2 kinase domain using FITC-KGGEEEEYFELVKK as substrate by peptide mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392008(CHEMBL2152398)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391996(CHEMBL2152300)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392018(CHEMBL2152409)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392003(CHEMBL2152307)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391990(CHEMBL2152296)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391990(CHEMBL2152296)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392001(CHEMBL2152305)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391986(CHEMBL2152422)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392010(CHEMBL2152400)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391989(CHEMBL2152424)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391991(CHEMBL2152425)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391996(CHEMBL2152300)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Inhibition of JAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391993(CHEMBL2152297)copy SMILEScopy InChI
Affinity DataKi:  4.20nMAssay Description:Inhibition of TYK2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  4.39nMAssay Description:Inhibition of human recombinant GST-tagged TYK2 using 5-FAM-KKSRGDYMTMQIG as substrate by peptide mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392001(CHEMBL2152305)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391984(CHEMBL2152420)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391996(CHEMBL2152300)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Inhibition of TYK2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392021(CHEMBL2152414)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391985(CHEMBL2152421)copy SMILEScopy InChI
Affinity DataKi:  5.90nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392019(CHEMBL2152412)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392020(CHEMBL2152413)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  7.80nMAssay Description:Inhibition of TYK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392017(CHEMBL2152408)copy SMILEScopy InChI
Affinity DataKi:  8.30nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391983(CHEMBL2152419)copy SMILEScopy InChI
Affinity DataKi:  9.30nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391987(CHEMBL2151053)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392007(CHEMBL2152397)copy SMILEScopy InChI
Affinity DataKi:  9.60nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391979(CHEMBL2152415)copy SMILEScopy InChI
Affinity DataKi:  9.80nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392015(CHEMBL2152406)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391982(CHEMBL2152418)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391995(CHEMBL2152299)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391980(CHEMBL2152416)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391988(CHEMBL2152423)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392013(CHEMBL2152404)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391999(CHEMBL2152303)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392005(CHEMBL2152395)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392004(CHEMBL2152394)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391995(CHEMBL2152299)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Inhibition of JAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50392014(CHEMBL2152405)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50391997(CHEMBL2152301)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KZXPubMed
Displayed 1 to 50 (of 127 total ) | Next | Last >>
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