Compile Data Set for Download or QSAR
Found 66 Enz. Inhib. hit(s) with all data for entry = 50040520
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395501(CHEMBL2163658)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Antagonist activity at KCNQ2/Q3 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395505(CHEMBL2164068)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM84184(2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide | 2...)copy SMILEScopy InChI
Affinity DataIC50: 163nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395508(CHEMBL2164062)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 4(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at KCNQ4 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395481(CHEMBL2163667)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395500(CHEMBL2163659)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395518(CHEMBL2164049)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395498(CHEMBL2163662)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395515(CHEMBL2164054)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395514(CHEMBL2164055)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395506(CHEMBL2164066)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395507(CHEMBL2164064)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395499(CHEMBL2163661)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395502(CHEMBL2163657)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395497(CHEMBL2163664)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395504(CHEMBL2164069)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM84166(2-phenyl-N-(2-phenylphenyl)butanamide | 2-phenyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395516(CHEMBL2164053)copy SMILEScopy InChI
Affinity DataIC50: 2.22E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 2.92E+3nMAssay Description:Antagonist activity at KCNQ1 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395503(CHEMBL2163655)copy SMILEScopy InChI
Affinity DataIC50: 3.31E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395517(CHEMBL2164052)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395475(CHEMBL2163350)copy SMILEScopy InChI
Affinity DataIC50: 5.27E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 8.12E+3nMAssay Description:Antagonist activity at KCNQ1/E1 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395479(CHEMBL2163673)copy SMILEScopy InChI
Affinity DataIC50: 1.27E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395474(CHEMBL2163686)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)copy SMILEScopy InChI
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395509(CHEMBL2164061)copy SMILEScopy InChI
Affinity DataIC50: 2.02E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395513(CHEMBL2164056)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395512(CHEMBL2164057)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395511(CHEMBL2164058)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395510(CHEMBL2164060)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395476(CHEMBL2163680)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395477(CHEMBL2163679)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395482(CHEMBL2163665)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395480(CHEMBL2163671)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395478(CHEMBL2163675)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395463(CHEMBL2163682)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395465(CHEMBL2163687)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395466(CHEMBL2163685)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395467(CHEMBL2163678)copy SMILEScopy InChI
Affinity DataEC50:  2.74E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395468(CHEMBL2163676)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395469(CHEMBL2163674)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395470(CHEMBL2163672)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395471(CHEMBL2163670)copy SMILEScopy InChI
Affinity DataEC50:  7.09E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2017PubMed
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