Compile Data Set for Download or QSAR
Found 9 Enz. Inhib. hit(s) with all data for entry = 50040802
TargetMetabotropic glutamate receptor 1(RAT)
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)copy SMILEScopy InChI
Affinity DataKi:  13.6nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400332(CHEMBL2181521)copy SMILEScopy InChI
Affinity DataKi:  22.2nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)copy SMILEScopy InChI
Affinity DataKi:  27.3nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)copy SMILEScopy InChI
Affinity DataIC50: 26.5nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400332(CHEMBL2181521)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)copy SMILEScopy InChI
Affinity DataIC50: 64.7nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGlu5 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400332(CHEMBL2181521)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGlu5 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGlu5 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7W5RPubMed