Compile Data Set for Download or QSAR
Found 68 Enz. Inhib. hit(s) with all data for entry = 50041853
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417006(CHEMBL1256414)copy SMILEScopy InChI
Affinity DataKi:  0.0790nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417006(CHEMBL1256414)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417006(CHEMBL1256414)copy SMILEScopy InChI
Affinity DataKi:  0.129nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417010(CHEMBL1255723)copy SMILEScopy InChI
Affinity DataKi:  0.138nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417010(CHEMBL1255723)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417019(CHEMBL1256378)copy SMILEScopy InChI
Affinity DataKi:  0.174nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417010(CHEMBL1255723)copy SMILEScopy InChI
Affinity DataKi:  0.182nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417019(CHEMBL1256378)copy SMILEScopy InChI
Affinity DataKi:  0.204nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417020(CHEMBL1256609)copy SMILEScopy InChI
Affinity DataKi:  0.219nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417019(CHEMBL1256378)copy SMILEScopy InChI
Affinity DataKi:  0.295nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417009(CHEMBL1255724)copy SMILEScopy InChI
Affinity DataKi:  0.347nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417009(CHEMBL1255724)copy SMILEScopy InChI
Affinity DataKi:  0.407nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417009(CHEMBL1255724)copy SMILEScopy InChI
Affinity DataKi:  0.437nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417008(CHEMBL1255771)copy SMILEScopy InChI
Affinity DataKi:  0.447nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417013(CHEMBL1256610)copy SMILEScopy InChI
Affinity DataKi:  0.513nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417020(CHEMBL1256609)copy SMILEScopy InChI
Affinity DataKi:  0.537nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417020(CHEMBL1256609)copy SMILEScopy InChI
Affinity DataKi:  0.692nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417012(CHEMBL1255616)copy SMILEScopy InChI
Affinity DataKi:  0.851nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417008(CHEMBL1255771)copy SMILEScopy InChI
Affinity DataKi:  0.912nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417018(CHEMBL1255770)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417018(CHEMBL1255770)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417018(CHEMBL1255770)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417013(CHEMBL1256610)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417012(CHEMBL1255616)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417021(CHEMBL1256566)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417013(CHEMBL1256610)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM81807(ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417011(CHEMBL1255617)copy SMILEScopy InChI
Affinity DataKi:  1.91nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417016(CHEMBL1256503)copy SMILEScopy InChI
Affinity DataKi:  1.95nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM81807(ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417012(CHEMBL1255616)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417008(CHEMBL1255771)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417016(CHEMBL1256503)copy SMILEScopy InChI
Affinity DataKi:  2.82nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417015(CHEMBL1256565)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417009(CHEMBL1255724)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-prazosin from human adrenergic alpha-1b receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417006(CHEMBL1256414)copy SMILEScopy InChI
Affinity DataKi:  3.55nMAssay Description:Displacement of [3H]-prazosin from human adrenergic alpha-1b receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417011(CHEMBL1255617)copy SMILEScopy InChI
Affinity DataKi:  3.89nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417021(CHEMBL1256566)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM81807(ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310)copy SMILEScopy InChI
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417020(CHEMBL1256609)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-prazosin from human adrenergic alpha-1b receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417021(CHEMBL1256566)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417007(FIPAMEZOLE)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417007(FIPAMEZOLE)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417012(CHEMBL1255616)copy SMILEScopy InChI
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]-prazosin from human adrenergic alpha-1b receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417015(CHEMBL1256565)copy SMILEScopy InChI
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417015(CHEMBL1256565)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417021(CHEMBL1256566)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-prazosin from human adrenergic alpha-1b receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417014(CHEMBL1256608)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417017(CHEMBL1256502)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417007(FIPAMEZOLE)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic Alpha-2C receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154X2PubMed
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