Affinity DataKd: 1.55E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 2.88E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.708nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.214nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 1.51E+4nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 5.75E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 6.31E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 158nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 8.71E+3nMAssay Description:Binding affinity to human recombinant sst3 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.32E+3nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 9.12E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.832nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.91E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.02E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 5.13E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.398nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 3.24E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.575nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.48E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.813nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.66E+4nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.407nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 3.55E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 5nMAssay Description:Binding affinity to human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 4.79E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 3.60nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 7.24E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 112nMAssay Description:Binding affinity to human 5HT1D receptorMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 224nMAssay Description:Binding affinity to human adrenergic beta-1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 7.90nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 1.78E+3nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 3.72E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 7.24E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Novartis Institutes for BioMedical Research
Curated by ChEMBL
Affinity DataKd: 3.63E+4nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 4.80nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair