Compile Data Set for Download or QSAR
Found 46 Enz. Inhib. hit(s) with all data for entry = 50042293
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423718(CHEMBL606371)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)copy SMILEScopy InChI
Affinity DataIC50: 257nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)copy SMILEScopy InChI
Affinity DataIC50: 261nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)copy SMILEScopy InChI
Affinity DataIC50: 319nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)copy SMILEScopy InChI
Affinity DataIC50: 347nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)copy SMILEScopy InChI
Affinity DataIC50: 472nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)copy SMILEScopy InChI
Affinity DataIC50: 502nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423718(CHEMBL606371)copy SMILEScopy InChI
Affinity DataIC50: 703nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)copy SMILEScopy InChI
Affinity DataIC50: 887nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)copy SMILEScopy InChI
Affinity DataIC50: 1.73E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)copy SMILEScopy InChI
Affinity DataIC50: 2.42E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)copy SMILEScopy InChI
Affinity DataIC50: 2.93E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)copy SMILEScopy InChI
Affinity DataIC50: 3.57E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)copy SMILEScopy InChI
Affinity DataIC50: 5.20E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)copy SMILEScopy InChI
Affinity DataIC50: 9.70E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)copy SMILEScopy InChI
Affinity DataIC50: 1.65E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)copy SMILEScopy InChI
Affinity DataIC50: 9.07E+4nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MKQPubMed