TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated lucifera...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inverse agonist activity at CCR4 in human HTLA cells assessed as depression of basal activity incubated for 20 mins by beta arrestin-recruitment medi...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruit...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated luciferase ...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruit...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inverse agonist activity at CCR4 in human HTLA cells assessed as depression of basal activity incubated for 20 mins by beta arrestin-recruitment medi...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inverse agonist activity at CCR4 in human HTLA cells assessed as depression of basal activity incubated for 20 mins by beta arrestin-recruitment medi...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated lucifera...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated lucifera...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruit...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated luciferase ...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated lucifera...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measured on day 4 by beta arr...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution me...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruit...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measured on day 4 by beta arrest...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by bet...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by beta a...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins measured on day 4 by beta arrestin-recruitment mediated luciferase ...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measured on day 4 by beta arr...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by beta a...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measure...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measure...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution me...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by bet...More data for this Ligand-Target Pair
TargetCruzipain(Trypanosoma cruzi)
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine using Z-Phe-Arg-aminomethylcoumarin as substrate incubated for 5 mins by spectrofluorimetric analysis in abs...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by bet...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of CX3CL1-stimulated CX3CR1 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by bet...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.78E+4nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measure...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of vasopressin-stimulated vasopressin V2 receptor in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution me...More data for this Ligand-Target Pair
TargetCruzipain(Trypanosoma cruzi)
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 8.27E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine using Z-Phe-Arg-aminomethylcoumarin as substrate incubated for 5 mins by spectrofluorimetric analysis in abs...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins with centrifuged compound solution measured on day 4 by beta arrest...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CCL22-stimulated CCR4 in human HTLA cells pre-incubated for 20 mins with Tween-80-treated compound solution measured on day 4 by beta a...More data for this Ligand-Target Pair
TargetCruzipain(Trypanosoma cruzi)
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine using Z-Phe-Arg-aminomethylcoumarin as substrate incubated for 5 mins by spectrofluorimetric analysis in pre...More data for this Ligand-Target Pair
TargetCruzipain(Trypanosoma cruzi)
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
University of North Carolina Chapel Hill School of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine using Z-Phe-Arg-aminomethylcoumarin as substrate incubated for 5 mins by spectrofluorimetric analysis in pre...More data for this Ligand-Target Pair