Compile Data Set for Download or QSAR
Found 53 Enz. Inhib. hit(s) with all data for entry = 50042944
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433573(CHEMBL2381570)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433565(CHEMBL2381567)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433570(CHEMBL2381571)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433568(CHEMBL2381564)copy SMILEScopy InChI
Affinity DataKi:  151nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433567(CHEMBL2381565)copy SMILEScopy InChI
Affinity DataKi:  217nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433571(CHEMBL2381569)copy SMILEScopy InChI
Affinity DataKi:  460nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)copy SMILEScopy InChI
Affinity DataKi:  6.70E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433570(CHEMBL2381571)copy SMILEScopy InChI
Affinity DataKi:  1.05E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433568(CHEMBL2381564)copy SMILEScopy InChI
Affinity DataKi:  2.93E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433565(CHEMBL2381567)copy SMILEScopy InChI
Affinity DataKi:  2.95E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433567(CHEMBL2381565)copy SMILEScopy InChI
Affinity DataKi:  4.87E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433571(CHEMBL2381569)copy SMILEScopy InChI
Affinity DataKi:  2.32E+5nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50241748(CHEMBL518059 | dihydro-beta-erythroidine)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50241748(CHEMBL518059 | dihydro-beta-erythroidine)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at (alpha4beta2)2alpha4 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433573(CHEMBL2381570)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433570(CHEMBL2381571)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433565(CHEMBL2381567)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50241748(CHEMBL518059 | dihydro-beta-erythroidine)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Antagonist activity at (alpha4beta2)2beta2 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curren...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433568(CHEMBL2381564)copy SMILEScopy InChI
Affinity DataIC50: 528nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433567(CHEMBL2381565)copy SMILEScopy InChI
Affinity DataIC50: 759nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433573(CHEMBL2381570)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at (alpha4beta2)2alpha4 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433571(CHEMBL2381569)copy SMILEScopy InChI
Affinity DataIC50: 1.61E+3nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at (alpha4beta2)2beta2 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curren...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Antagonist activity at (alpha4beta2)2beta2 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curren...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Antagonist activity at (alpha4beta2)2alpha4 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433573(CHEMBL2381570)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Antagonist activity at (alpha4beta2)2beta2 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curren...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataIC50: 1.78E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433570(CHEMBL2381571)copy SMILEScopy InChI
Affinity DataIC50: 2.11E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)copy SMILEScopy InChI
Affinity DataIC50: 2.58E+4nMAssay Description:Antagonist activity at (alpha4beta2)2beta2 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curren...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)copy SMILEScopy InChI
Affinity DataIC50: 5.23E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433568(CHEMBL2381564)copy SMILEScopy InChI
Affinity DataIC50: 5.85E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433565(CHEMBL2381567)copy SMILEScopy InChI
Affinity DataIC50: 5.91E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)copy SMILEScopy InChI
Affinity DataIC50: 9.50E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha4 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile

Curated by ChEMBL
LigandPNGBDBM50433567(CHEMBL2381565)copy SMILEScopy InChI
Affinity DataIC50: 9.73E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2JJQPubMed
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