Compile Data Set for Download or QSAR
Found 72 Enz. Inhib. hit(s) with all data for entry = 50042983
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434163(CHEMBL2385273 | US9346814, Cmpd No 12 Example 15)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434164(CHEMBL2385272 | US9346814, Cmpd No 13 Example 16)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434165(CHEMBL2385271 | US9346814, Cmpd No 11 Example 14)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434170(CHEMBL2385299 | US9346814, Cmpd No 21 Example 25)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434166(CHEMBL2385270 | US9346814, Cmpd No 6 Example 9)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434167(CHEMBL2385302 | US9346814, Cmpd No 8 Example 11)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434168(CHEMBL2385301 | US9346814, Cmpd No 7 Example 10)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434191(CHEMBL2385278)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434190(CHEMBL2385279)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434171(CHEMBL2385298 | US9346814, Cmpd No 38 Example 43)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434162(CHEMBL2385274 | US9346814, Cmpd No 9 Example 12)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434174(CHEMBL2385295)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434162(CHEMBL2385274 | US9346814, Cmpd No 9 Example 12)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434161(CHEMBL2385275 | US9346814, Cmpd No 10 Example 13)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434161(CHEMBL2385275 | US9346814, Cmpd No 10 Example 13)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434159(CHEMBL2385277 | US9346814, Ref Cmpd No 7 (example ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434183(CHEMBL2385286)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434160(CHEMBL2385276)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434166(CHEMBL2385270 | US9346814, Cmpd No 6 Example 9)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434176(CHEMBL2385293 | US9346814, Cmpd No 3 Example 4)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434176(CHEMBL2385293 | US9346814, Cmpd No 3 Example 4)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434167(CHEMBL2385302 | US9346814, Cmpd No 8 Example 11)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434172(CHEMBL2385297)copy SMILEScopy InChI
Affinity DataIC50: 770nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434168(CHEMBL2385301 | US9346814, Cmpd No 7 Example 10)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434173(CHEMBL2385296)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434174(CHEMBL2385295)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434163(CHEMBL2385273 | US9346814, Cmpd No 12 Example 15)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434164(CHEMBL2385272 | US9346814, Cmpd No 13 Example 16)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434178(CHEMBL2385291)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434189(CHEMBL2385280 | US9346814, Ref. Cmpd No 6 (Example...)copy SMILEScopy InChI
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434178(CHEMBL2385291)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434191(CHEMBL2385278)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434159(CHEMBL2385277 | US9346814, Ref Cmpd No 7 (example ...)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434187(CHEMBL2385282)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434160(CHEMBL2385276)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434184(CHEMBL2385285)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434175(CHEMBL2385294 | US9346814, Cmpd No 5 Example 8)copy SMILEScopy InChI
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434165(CHEMBL2385271 | US9346814, Cmpd No 11 Example 14)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434185(CHEMBL2385284)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434189(CHEMBL2385280 | US9346814, Ref. Cmpd No 6 (Example...)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434180(CHEMBL2385289)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434183(CHEMBL2385286)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
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