Compile Data Set for Download or QSAR
Found 98 Enz. Inhib. hit(s) with all data for entry = 50043118
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436256(CHEMBL2398726)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436283(CHEMBL2398729)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436256(CHEMBL2398726)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of RANTES-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436260(CHEMBL2398717)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436288(CHEMBL2398728)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436287(CHEMBL2398744)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436282(CHEMBL2398769)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436284(CHEMBL2398747 | US8633226, 460)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436288(CHEMBL2398728)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436308(CHEMBL2398739)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436287(CHEMBL2398744)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436307(CHEMBL2398746)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436286(CHEMBL2398737)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436285(CHEMBL2398743 | US8633226, 466)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436256(CHEMBL2398726)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436306(CHEMBL2398748)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436257(CHEMBL2398724)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436258(CHEMBL2398722)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436276(CHEMBL2398750)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436284(CHEMBL2398747 | US8633226, 460)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436305(CHEMBL2398749)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436256(CHEMBL2398726)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MPIF-1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436270(CHEMBL2398763)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436283(CHEMBL2398729)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436285(CHEMBL2398743 | US8633226, 466)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436274(CHEMBL2398767)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436304(CHEMBL2398745)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436258(CHEMBL2398722)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436278(CHEMBL2398730)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436264(CHEMBL2398765)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436282(CHEMBL2398769)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436281(CHEMBL2398741)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436266(CHEMBL2398757)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436256(CHEMBL2398726)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of HCC-1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436268(CHEMBL2398758)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436286(CHEMBL2398737)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436277(CHEMBL2398735)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436256(CHEMBL2398726)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of ieukotactin-1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436280(CHEMBL2398742)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436281(CHEMBL2398741)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436280(CHEMBL2398742)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436279(CHEMBL2398770)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436259(CHEMBL2398716 | US8633226, 1356)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436278(CHEMBL2398730)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436257(CHEMBL2398724)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436303(CHEMBL2398738)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436277(CHEMBL2398735)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436271(CHEMBL2398727)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436279(CHEMBL2398770)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50436261(CHEMBL2398764)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X596GPubMed
Displayed 1 to 50 (of 98 total ) | Next | Last >>
Jump to: