TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by double-reciprocal plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of human matriptase measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human matriptase measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-14(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-14(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-14(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human matriptase measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human matriptase measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human matriptase measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-14(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
TargetKallikrein-14(Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair