Found 9 Enz. Inhib. hit(s) with all data for entry = 50043494 TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
3D Structure (crystal)TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 311nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 402nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 1.63E+3nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 2.44E+3nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 2.57E+3nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Activity at human MDR1 expressed in MDCK cells assessed as Calcein-AM uptake after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Universit£ degli Studi di Bari ALDO MORO
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Activity at human MDR1 expressed in MDCK cells assessed as Calcein-AM uptake after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
