Compile Data Set for Download or QSAR
Found 17 Enz. Inhib. hit(s) with all data for entry = 50043627
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443803(CHEMBL3094250)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443800(CHEMBL3094255)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443805(CHEMBL3094249)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM81395(APO-866)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443801(CHEMBL3094254)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443798(CHEMBL3094258)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443799(CHEMBL3094257)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443796(CHEMBL3094229)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443802(CHEMBL3094251)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443793(CHEMBL3094236)copy SMILEScopy InChI
Affinity DataIC50: 8.20nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443791(CHEMBL3094238)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50435350(CHEMBL17289)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443797(CHEMBL3094224)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443804(CHEMBL2417795)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443794(CHEMBL3094234)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443795(CHEMBL3094230)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Topotarget A/S

Curated by ChEMBL
LigandPNGBDBM50443792(CHEMBL3094237)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:Inhibition of NAMPT in human HepG2 cells using [14C]-nicotinamide/PRPP as substrate assessed as formation of [14C]-nicotinamide mononucleotide after ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4K6WPubMed