Compile Data Set for Download or QSAR
Found 36 Enz. Inhib. hit(s) with all data for entry = 50044186
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008271(CHEMBL3235132)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human TAF1a using hippuryl-L-arginine/hippuryl-L-lysine as substrate by liquid chromatographic analysisMore data for this Ligand-Target Pair
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008272(CHEMBL3235133)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008279(CHEMBL3235140)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008278(CHEMBL3235139)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008271(CHEMBL3235132)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008273(CHEMBL3235134)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008269(CHEMBL3235130)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of human TAF1a using hippuryl-L-arginine/hippuryl-L-lysine as substrate by liquid chromatographic analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008272(CHEMBL3235133)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008274(CHEMBL3235135)copy SMILEScopy InChI
Affinity DataIC50: 106nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008273(CHEMBL3235134)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008275(CHEMBL3235136)copy SMILEScopy InChI
Affinity DataIC50: 124nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008269(CHEMBL3235130)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50226610((2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibition of human TAF1a using hippuryl-L-arginine/hippuryl-L-lysine as substrate by liquid chromatographic analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008276(CHEMBL3235137)copy SMILEScopy InChI
Affinity DataIC50: 585nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008270(CHEMBL3235131)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of human TAF1a using hippuryl-L-arginine/hippuryl-L-lysine as substrate by liquid chromatographic analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008271(CHEMBL3235132)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008278(CHEMBL3235139)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50135933(3-(6-Amino-pyridin-3-yl)-2-(1H-imidazol-4-yl)-prop...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human TAF1a using hippuryl-L-arginine/hippuryl-L-lysine as substrate by liquid chromatographic analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008277(CHEMBL3235138)copy SMILEScopy InChI
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of human TAF1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008274(CHEMBL3235135)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008279(CHEMBL3235140)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50226610((2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008276(CHEMBL3235137)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008270(CHEMBL3235131)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008275(CHEMBL3235136)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50135933(3-(6-Amino-pyridin-3-yl)-2-(1H-imidazol-4-yl)-prop...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008277(CHEMBL3235138)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TAF1a in human plasma assessed as clot lysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008277(CHEMBL3235138)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008278(CHEMBL3235139)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008276(CHEMBL3235137)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008275(CHEMBL3235136)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008274(CHEMBL3235135)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008273(CHEMBL3235134)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008279(CHEMBL3235140)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008271(CHEMBL3235132)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50008272(CHEMBL3235133)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of carboxypeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09TGPubMed