TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.0680nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.630nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]2-iodomelatonin from MT1 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Antagonist activity at human MT2 receptorMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [125I]2-iodomelatonin from MT1 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Antagonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Displacement of [125I]2-iodomelatonin from MT1 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 87nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair