Compile Data Set for Download or QSAR
Found 52 Enz. Inhib. hit(s) with all data for entry = 50044533
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020015(CHEMBL3287814)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020014(CHEMBL3287813)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020011(CHEMBL3287810)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020011(CHEMBL3287810)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020015(CHEMBL3287814)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019982(CHEMBL3287584)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020012(CHEMBL3287811)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019983(CHEMBL3287585)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019983(CHEMBL3287585)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020012(CHEMBL3287811)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020010(CHEMBL3287586)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020014(CHEMBL3287813)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020010(CHEMBL3287586)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020013(CHEMBL3287812)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019982(CHEMBL3287584)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019979(CHEMBL3287833)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020020(CHEMBL3287819)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020022(CHEMBL3287821)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019979(CHEMBL3287833)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019976(CHEMBL3287827)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020020(CHEMBL3287819)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020022(CHEMBL3287821)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019974(CHEMBL3287825)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019977(CHEMBL3287828)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019973(CHEMBL3287824)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019976(CHEMBL3287827)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019980(CHEMBL3287834)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019975(CHEMBL3287826)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020019(CHEMBL3287818)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020024(CHEMBL3287829)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019984(CHEMBL528724 | GNF-Pf-1241)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019978(CHEMBL3287832)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019974(CHEMBL3287825)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019981(CHEMBL3287835)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020018(CHEMBL3287817)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019977(CHEMBL3287828)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019973(CHEMBL3287824)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019984(CHEMBL528724 | GNF-Pf-1241)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020016(CHEMBL3287815)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020021(CHEMBL3287820)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019980(CHEMBL3287834)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019981(CHEMBL3287835)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019975(CHEMBL3287826)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019978(CHEMBL3287832)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019972(CHEMBL3287823)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020018(CHEMBL3287817)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020026(CHEMBL3287831)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020021(CHEMBL3287820)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50019972(CHEMBL3287823)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50020017(CHEMBL3287816)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+4nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V989NRPubMed
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