Compile Data Set for Download or QSAR
Found 256 Enz. Inhib. hit(s) with all data for entry = 50045163
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)copy SMILEScopy InChI
Affinity DataKi:  0.0480nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50109461(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047991(CHEMBL3314888)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047979(CHEMBL3314876)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047990(CHEMBL3314887)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047986(CHEMBL3314883)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047980(CHEMBL3314877)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047995(CHEMBL3314892)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047993(CHEMBL3314890)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048011(CHEMBL3314895)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047992(CHEMBL3314889)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047978(CHEMBL3313941)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047982(CHEMBL3314879)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048020(CHEMBL3314903)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047977(CHEMBL3314875)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048031(CHEMBL3314913)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048060(CHEMBL3314873)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047985(CHEMBL3314882)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048020(CHEMBL3314903)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048011(CHEMBL3314895)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047996(CHEMBL3314893)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047996(CHEMBL3314893)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047995(CHEMBL3314892)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047994(CHEMBL3314891)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048058(CHEMBL3314871)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048014(CHEMBL3314898)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047993(CHEMBL3314890)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047997(CHEMBL3314894)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047996(CHEMBL3314893)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048031(CHEMBL3314913)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048031(CHEMBL3314913)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048014(CHEMBL3314898)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047992(CHEMBL3314889)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047991(CHEMBL3314888)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047983(CHEMBL3314880)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048012(CHEMBL3314896)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047978(CHEMBL3313941)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048015(CHEMBL3314899)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048013(CHEMBL3314897)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048029(CHEMBL3314911)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047995(CHEMBL3314892)copy SMILEScopy InChI
Affinity DataKi:  61nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048061(CHEMBL3314874)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048015(CHEMBL3314899)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048020(CHEMBL3314903)copy SMILEScopy InChI
Affinity DataKi:  75nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048061(CHEMBL3314874)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047993(CHEMBL3314890)copy SMILEScopy InChI
Affinity DataKi:  103nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50047990(CHEMBL3314887)copy SMILEScopy InChI
Affinity DataKi:  104nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048026(CHEMBL3314908)copy SMILEScopy InChI
Affinity DataKi:  105nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£ di Trieste

Curated by ChEMBL
LigandPNGBDBM50048058(CHEMBL3314871)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NPSPubMed
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