Compile Data Set for Download or QSAR
Found 94 Enz. Inhib. hit(s) with all data for entry = 50045710
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078007(CHEMBL3417384)copy SMILES
Affinity DataKi:  0.0160nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077994(CHEMBL3417378)copy SMILES
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078002(CHEMBL3417389)copy SMILES
Affinity DataKi:  0.340nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078006(CHEMBL3417385)copy SMILES
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077995(CHEMBL3417377)copy SMILES
Affinity DataKi:  0.480nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078001(CHEMBL3417390)copy SMILES
Affinity DataKi:  0.690nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077993(CHEMBL3417379)copy SMILES
Affinity DataKi:  1nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078005(CHEMBL3417386)copy SMILES
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077992(CHEMBL3417380)copy SMILES
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078000(CHEMBL3414601)copy SMILES
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077999(CHEMBL3417291)copy SMILES
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078003(CHEMBL3417388)copy SMILES
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078010(CHEMBL3417381)copy SMILES
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078008(CHEMBL3417383)copy SMILES
Affinity DataKi:  5.40nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077997(CHEMBL3417375)copy SMILES
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077998(CHEMBL3414600)copy SMILES
Affinity DataKi:  9.10nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078004(CHEMBL3417387)copy SMILES
Affinity DataKi:  11nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078009(CHEMBL3417382)copy SMILES
Affinity DataKi:  11nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077996(CHEMBL3417376)copy SMILES
Affinity DataKi:  15nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078014(CHEMBL3417391)copy SMILES
Affinity DataKi:  46nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078013(CHEMBL3417392)copy SMILES
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078011(CHEMBL3417394)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078012(CHEMBL3417393)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078007(CHEMBL3417384)copy SMILES
Affinity DataIC50: 0.0200nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077994(CHEMBL3417378)copy SMILES
Affinity DataIC50: 0.25nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078002(CHEMBL3417389)copy SMILES
Affinity DataIC50: 0.430nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078006(CHEMBL3417385)copy SMILES
Affinity DataIC50: 0.480nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077995(CHEMBL3417377)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078001(CHEMBL3417390)copy SMILES
Affinity DataIC50: 0.860nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077993(CHEMBL3417379)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078005(CHEMBL3417386)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077992(CHEMBL3417380)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078000(CHEMBL3414601)copy SMILES
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077999(CHEMBL3417291)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078003(CHEMBL3417388)copy SMILES
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078010(CHEMBL3417381)copy SMILES
Affinity DataIC50: 6.10nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078008(CHEMBL3417383)copy SMILES
Affinity DataIC50: 6.70nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077997(CHEMBL3417375)copy SMILES
Affinity DataIC50: 7.90nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077998(CHEMBL3414600)copy SMILES
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078009(CHEMBL3417382)copy SMILES
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078004(CHEMBL3417387)copy SMILES
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50077996(CHEMBL3417376)copy SMILES
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078014(CHEMBL3417391)copy SMILES
Affinity DataIC50: 57nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078011(CHEMBL3417394)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078012(CHEMBL3417393)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078013(CHEMBL3417392)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078002(CHEMBL3417389)copy SMILES
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human APJ receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced intracellular cAMP production incubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£ de Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50078003(CHEMBL3417388)copy SMILES
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human APJ receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced intracellular cAMP production incubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GNRPubMed
Displayed 1 to 50 (of 94 total ) | Next | Last >>
Jump to: