Found 7 Enz. Inhib. hit(s) with all data for entry = 50045947 TargetSolute carrier family 22 member 6(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 4.51E+7nMAssay Description:Binding affinity to human OAT1More data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+7nMAssay Description:Inhibition of mouse recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation...More data for this Ligand-Target Pair
Affinity DataIC50: 1.83E+7nMAssay Description:Inhibition of rat recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation c...More data for this Ligand-Target Pair
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.74E+7nMAssay Description:Inhibition of human recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation...More data for this Ligand-Target Pair
Affinity DataKd: 2.20nMAssay Description:Activity at mouse recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scint...More data for this Ligand-Target Pair
Affinity DataKd: 2.20nMAssay Description:Activity at rat recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scintil...More data for this Ligand-Target Pair
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKd: 2.20nMAssay Description:Activity at human recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scint...More data for this Ligand-Target Pair
