Compile Data Set for Download or QSAR
Found 66 Enz. Inhib. hit(s) with all data for entry = 50046051
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092784(CHEMBL3586382)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092785(CHEMBL3586383)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092786(CHEMBL3586384)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50431521(CHEMBL2348864)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092783(CHEMBL3586404)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092769(CHEMBL3586397)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092782(CHEMBL3586387)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092780(CHEMBL3586385)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092793(CHEMBL3586380)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092783(CHEMBL3586404)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of cFMS (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092783(CHEMBL3586404)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092787(CHEMBL3585359)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092766(CHEMBL3586401)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092773(CHEMBL3586394)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092789(CHEMBL3586405)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant mTOR (unknown origin) using GST-p70S6 as substrate after 60 mins by TR-FRET analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092792(CHEMBL3586379)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092791(CHEMBL3586389)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092781(CHEMBL3586386)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092771(CHEMBL3586399)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092784(CHEMBL3586382)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092768(CHEMBL3586403)copy SMILEScopy InChI
Affinity DataIC50: 103nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092788(CHEMBL3586381)copy SMILEScopy InChI
Affinity DataIC50: 103nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50431519(CHEMBL2348862)copy SMILEScopy InChI
Affinity DataIC50: 106nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092774(CHEMBL3586395)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092786(CHEMBL3586384)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092790(CHEMBL3586388)copy SMILEScopy InChI
Affinity DataIC50: 122nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092775(CHEMBL3586396)copy SMILEScopy InChI
Affinity DataIC50: 149nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092777(CHEMBL3586393)copy SMILEScopy InChI
Affinity DataIC50: 168nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092770(CHEMBL3586398)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092779(CHEMBL3586391)copy SMILEScopy InChI
Affinity DataIC50: 175nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092776(CHEMBL3586392)copy SMILEScopy InChI
Affinity DataIC50: 185nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092773(CHEMBL3586394)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092785(CHEMBL3586383)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092772(CHEMBL3586400)copy SMILEScopy InChI
Affinity DataIC50: 203nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092770(CHEMBL3586398)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092787(CHEMBL3585359)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092788(CHEMBL3586381)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092767(CHEMBL3586402)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092768(CHEMBL3586403)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50431519(CHEMBL2348862)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092778(CHEMBL3586390)copy SMILEScopy InChI
Affinity DataIC50: 436nMAssay Description:Inhibition of mTOR (unknown origin) by HTR-FRET substrate phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092782(CHEMBL3586387)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092767(CHEMBL3586402)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50431521(CHEMBL2348864)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetFKBP12A/mTOR(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092779(CHEMBL3586391)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as inhibition of S6 phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092783(CHEMBL3586404)copy SMILEScopy InChI
Affinity DataIC50: 651nMAssay Description:Inhibition of Flt4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092780(CHEMBL3586385)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092766(CHEMBL3586401)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092781(CHEMBL3586386)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50092769(CHEMBL3586397)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PI3K-alpha (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208672FPubMed
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