Compile Data Set for Download or QSAR
Found 24 Enz. Inhib. hit(s) with all data for entry = 50046103
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094926(CHEMBL3589282)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094927(CHEMBL3589283)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094926(CHEMBL3589282)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094941(CHEMBL3589285)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094927(CHEMBL3589283)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50318567(2-(4-(Trifluoromethyl)phenyl)-7,8-dihydro-5H-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50318567(2-(4-(Trifluoromethyl)phenyl)-7,8-dihydro-5H-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094928(CHEMBL3589284)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094925(CHEMBL3589281)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094928(CHEMBL3589284)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094925(CHEMBL3589281)copy SMILEScopy InChI
Affinity DataIC50: 189nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094924(CHEMBL3589258)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094941(CHEMBL3589285)copy SMILEScopy InChI
Affinity DataIC50: 423nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094925(CHEMBL3589281)copy SMILEScopy InChI
Affinity DataIC50: 949nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094923(CHEMBL3589254)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094941(CHEMBL3589285)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094928(CHEMBL3589284)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094923(CHEMBL3589254)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094926(CHEMBL3589282)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094927(CHEMBL3589283)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094922(CHEMBL3589247)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094924(CHEMBL3589258)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094922(CHEMBL3589247)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of human TNKS2 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50094924(CHEMBL3589258)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35072PubMed