Affinity DataKi: 4.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.91E+3nMAssay Description:Inhibition of PGM1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.78E+4nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Homo sapiens (Human))
Universit£ di Pisa
Curated by ChEMBL
Universit£ di Pisa
Curated by ChEMBL
Affinity DataIC50: 207nMAssay Description:Inhibition of PFKFB3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of hexokinase 2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 576nMAssay Description:Inhibition of ENO1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of LDHB (unknown origin)More data for this Ligand-Target Pair
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Homo sapiens (Human))
Universit£ di Pisa
Curated by ChEMBL
Universit£ di Pisa
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of PFKFB3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of LDHA (unknown origin) by pyruvate competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of PGM1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of LDHA (unknown origin) by NADH competition assayMore data for this Ligand-Target Pair
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Homo sapiens (Human))
Universit£ di Pisa
Curated by ChEMBL
Universit£ di Pisa
Curated by ChEMBL
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of PFKFB3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Binding affinity to MCT1 (unknown origin)More data for this Ligand-Target Pair