Compile Data Set for Download or QSAR
Found 9 Enz. Inhib. hit(s) with all data for entry = 50046337
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106623(CHEMBL3600871)copy SMILEScopy InChI
Affinity DataKd:  0.440nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106624(CHEMBL3600870)copy SMILEScopy InChI
Affinity DataKd:  0.730nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106625(CHEMBL3600869)copy SMILEScopy InChI
Affinity DataKd:  2.5nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106626(CHEMBL3600868)copy SMILEScopy InChI
Affinity DataKd:  6.10nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106631(CHEMBL3600653)copy SMILEScopy InChI
Affinity DataKd:  1.90nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106628(CHEMBL3600763)copy SMILEScopy InChI
Affinity DataKd:  6.5nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106629(CHEMBL3600762)copy SMILEScopy InChI
Affinity DataKd:  9.10nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106630(CHEMBL3600760)copy SMILEScopy InChI
Affinity DataKd:  2.20nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50106627(CHEMBL3600764)copy SMILEScopy InChI
Affinity DataKd:  5.70nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NMTPubMed