Compile Data Set for Download or QSAR
Found 71 Enz. Inhib. hit(s) with all data for entry = 50047157
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150818(CHEMBL3774575)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150821(CHEMBL3775251)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150820(CHEMBL3774933)copy SMILEScopy InChI
Affinity DataIC50: 8.30nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150758(CHEMBL3775901)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150822(CHEMBL3775348)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150756(CHEMBL3774766)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150819(CHEMBL3774542)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150812(CHEMBL3775853 | US10702504, Compound D)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150811(CHEMBL3775073)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150808(CHEMBL3774507 | US10702504, Compound C)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150757(CHEMBL3774770)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150761(CHEMBL3775689)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150801(CHEMBL3775132)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150796(CHEMBL3774529)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150815(CHEMBL3775263)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150759(CHEMBL3774638)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150803(CHEMBL3774452)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150813(CHEMBL3774653)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150816(CHEMBL3775286)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150814(CHEMBL3775640)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150760(CHEMBL3774883)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50148479(CHEMBL3770259)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150824(CHEMBL3775297)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150817(CHEMBL3774616)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150800(CHEMBL3775687)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150874(CHEMBL3775559)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150872(CHEMBL3774404)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150873(CHEMBL3774673)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150825(CHEMBL3774804)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150876(CHEMBL3775715)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150828(CHEMBL3774650)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150908(CHEMBL3775440)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of KDM3A (unknown origin) using biotin-H3K9me2 (1 to 21 residues) as substrate preincubated for 15 mins followed by substrate addition mea...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150827(CHEMBL1557110)copy SMILEScopy InChI
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150823(CHEMBL1365878)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150881(CHEMBL3775616)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150907(CHEMBL3774967)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150826(CHEMBL1734009)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150871(CHEMBL3775315)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate preincubated for 15 mins followed by substrate addition m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150756(CHEMBL3774766)copy SMILEScopy InChI
Affinity DataEC50:  170nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150757(CHEMBL3774770)copy SMILEScopy InChI
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150758(CHEMBL3775901)copy SMILEScopy InChI
Affinity DataEC50:  170nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150759(CHEMBL3774638)copy SMILEScopy InChI
Affinity DataEC50:  5.50E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150760(CHEMBL3774883)copy SMILEScopy InChI
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150761(CHEMBL3775689)copy SMILEScopy InChI
Affinity DataEC50:  1.90E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150796(CHEMBL3774529)copy SMILEScopy InChI
Affinity DataEC50:  2.70E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150800(CHEMBL3775687)copy SMILEScopy InChI
Affinity DataEC50: >3.60E+4nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150801(CHEMBL3775132)copy SMILEScopy InChI
Affinity DataEC50:  5.00E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150803(CHEMBL3774452)copy SMILEScopy InChI
Affinity DataEC50:  3.00E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150808(CHEMBL3774507 | US10702504, Compound C)copy SMILEScopy InChI
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150811(CHEMBL3775073)copy SMILEScopy InChI
Affinity DataEC50:  950nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26975F4PubMed
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