Compile Data Set for Download or QSAR
Found 69 Enz. Inhib. hit(s) with all data for entry = 50047306
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-Angiotensin 2 from human placental AT1 receptor expressed in African green monkey COS7 cell membranes after 90 mins by gamma cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)copy SMILEScopy InChI
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159160(CHEMBL3786779)copy SMILEScopy InChI
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159205(CHEMBL3785233)copy SMILEScopy InChI
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159164(CHEMBL3787200)copy SMILEScopy InChI
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159155(CHEMBL3786852)copy SMILEScopy InChI
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159156(CHEMBL3786291)copy SMILEScopy InChI
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159232(CHEMBL3786263)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of S0586[K4]hpp from human NPY4 receptor expressed in CHO cells co-expressing Gqi5-mtAEQ by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159227(CHEMBL3786309)copy SMILEScopy InChI
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]EYE from human NPFF2 receptor expressed in CHO cell membranes after 1 hr by liquid scintillation spectrophotometric countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159212(CHEMBL3786771)copy SMILEScopy InChI
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159156(CHEMBL3786291)copy SMILEScopy InChI
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from human NTSR1 transfec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159155(CHEMBL3786852)copy SMILEScopy InChI
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from human NTSR1 transfec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159153(CHEMBL3787243)copy SMILEScopy InChI
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159155(CHEMBL3786852)copy SMILEScopy InChI
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]NT(8 to 13 residues) from human NTSR2 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]EYE from human NPFF2 receptor expressed in CHO cell membranes after 1 hr by liquid scintillation spectrophotometric countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]NT(8 to 13 residues) from human NTSR2 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159230(CHEMBL3785569)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of S0586[K4]hpp from human NPY4 receptor expressed in CHO cells co-expressing Gqi5-mtAEQ by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159183(CHEMBL3787095)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159212(CHEMBL3786771)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from human NTSR1 transfec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159151(CHEMBL3786145)copy SMILEScopy InChI
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159156(CHEMBL3786291)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]NT(8 to 13 residues) from human NTSR2 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159152(CHEMBL3786986)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159154(CHEMBL3787379)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50240609(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159231(CHEMBL3787528)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of S0586[K4]hpp from human NPY4 receptor expressed in CHO cells co-expressing Gqi5-mtAEQ by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159186(CHEMBL3786135)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159228(CHEMBL3785576)copy SMILEScopy InChI
Affinity DataKi:  7.40nMAssay Description:Displacement of S0586[K4]hpp from human NPY4 receptor expressed in CHO cells co-expressing Gqi5-mtAEQ by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159186(CHEMBL3786135)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from human NTSR1 transfec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159157(CHEMBL3785563)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159159(CHEMBL3786195)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-Angiotensin 2 from AT1 receptor in human PLC/PRF/5 cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159225(CHEMBL3786583)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H]EYE from human NPFF2 receptor expressed in CHO cell membranes after 1 hr by liquid scintillation spectrophotometric countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159226(CHEMBL3786376)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Displacement of [3H]EYE from human NPFF2 receptor expressed in CHO cell membranes after 1 hr by liquid scintillation spectrophotometric countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)copy SMILEScopy InChI
Affinity DataIC50: 0.407nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50240609(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:Displacement of [3H]-Angiotensin 2 from human AT1 receptor transfected in CHOK1 cells preincubated for 30 mins with bovine serum albumin followed by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)copy SMILEScopy InChI
Affinity DataIC50: 0.724nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159155(CHEMBL3786852)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159156(CHEMBL3786291)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159212(CHEMBL3786771)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159153(CHEMBL3787243)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159183(CHEMBL3787095)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-Arg-ProTyr-Ile-Leu-OH Tris(hydrotrifluoroacetate) from NTSR1 in human HT-29...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159151(CHEMBL3786145)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50240609(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159157(CHEMBL3785563)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]-Asp-{Nomega-[N-(4-propanoylaminobutyl)aminocarbonyl]}Arg-ValTyr-Ile-His-Pro-Phe-OH Tris(hydrotrifluoroacetate) from human AT1 re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159154(CHEMBL3787379)copy SMILEScopy InChI
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159153(CHEMBL3787243)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69MGKPubMed
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