Compile Data Set for Download or QSAR
Found 92 Enz. Inhib. hit(s) with all data for entry = 50047409
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102978(US8546435, 6)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165587(CHEMBL3800298)copy SMILEScopy InChI
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102979(US8546435, 7)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165582(CHEMBL3797225)copy SMILEScopy InChI
Affinity DataKi:  2.5nM ΔG°:  -49.1kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165589(CHEMBL3798095)copy SMILEScopy InChI
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165588(CHEMBL3800422)copy SMILEScopy InChI
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165592(CHEMBL3799776)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102977(US8546435, 5)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165583(CHEMBL3798645)copy SMILEScopy InChI
Affinity DataKi:  8nM ΔG°:  -46.2kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165590(CHEMBL3799225)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102975(US8546435, 3)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102976(US8546435, 4)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165591(CHEMBL3798155)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102980(US8546435, 8)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165593(CHEMBL3799687)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165581(CHEMBL3799222)copy SMILEScopy InChI
Affinity DataKi:  17nM ΔG°:  -44.3kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165594(CHEMBL3797531)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165586(CHEMBL3798559)copy SMILEScopy InChI
Affinity DataKi:  30nM ΔG°:  -42.9kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102981(US8546435, 9)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165596(CHEMBL3798525)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165585(CHEMBL3800172)copy SMILEScopy InChI
Affinity DataKi:  50nM ΔG°:  -41.7kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165598(CHEMBL3797857)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165595(CHEMBL3799883)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165601(CHEMBL3799671)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165584(CHEMBL3798056)copy SMILEScopy InChI
Affinity DataKi:  110nM ΔG°:  -39.7kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165604(CHEMBL3798204)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165599(CHEMBL3799862)copy SMILEScopy InChI
Affinity DataKi:  154nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165602(CHEMBL3799604)copy SMILEScopy InChI
Affinity DataKi:  154nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165579(CHEMBL3797639)copy SMILEScopy InChI
Affinity DataKi:  210nM ΔG°:  -38.1kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165580(CHEMBL3798337)copy SMILEScopy InChI
Affinity DataKi:  220nM ΔG°:  -38.0kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50260270(CHEMBL506986 | KwFwLL-NH2)copy SMILEScopy InChI
Affinity DataKi:  255nM ΔG°:  -37.6kJ/moleT: 2°CAssay Description:Competitive binding affinity to human SNAP-tagged GHS-R1a expressed in HEK293T cells incubated at 4 degC for 3 hrs or at room temperature for 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165600(CHEMBL3799567)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165605(CHEMBL3800383)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165597(CHEMBL3800225)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165603(CHEMBL3800176)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165592(CHEMBL3799776)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102976(US8546435, 4)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102978(US8546435, 6)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165592(CHEMBL3799776)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102975(US8546435, 3)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102975(US8546435, 3)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102977(US8546435, 5)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165590(CHEMBL3799225)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102979(US8546435, 7)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165591(CHEMBL3798155)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165591(CHEMBL3798155)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165594(CHEMBL3797531)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165590(CHEMBL3799225)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM102976(US8546435, 4)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier

Curated by ChEMBL
LigandPNGBDBM50165594(CHEMBL3797531)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9688VPubMed
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