Compile Data Set for Download or QSAR
Found 124 Enz. Inhib. hit(s) with all data for entry = 50047692
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183567(CHEMBL3823177)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183568(CHEMBL3823369)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183561(CHEMBL3824146)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183453(CHEMBL3824312)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183562(CHEMBL3823599)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183562(CHEMBL3823599)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183563(CHEMBL3823697)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183561(CHEMBL3824146)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of human BRD7 measured after mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183517(CHEMBL3823859 | US11773085, Compound B50)copy SMILEScopy InChI
Affinity DataIC50: 128nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183452(CHEMBL3824351)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183450(CHEMBL3824133)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183454(CHEMBL3822539)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183453(CHEMBL3824312)copy SMILEScopy InChI
Affinity DataIC50: 188nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183570(CHEMBL3824289)copy SMILEScopy InChI
Affinity DataIC50: 195nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183563(CHEMBL3823697)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183560(CHEMBL3822909)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183569(CHEMBL3823906)copy SMILEScopy InChI
Affinity DataIC50: 468nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183572(CHEMBL3822988)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183451(CHEMBL3823551)copy SMILEScopy InChI
Affinity DataIC50: 507nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183571(CHEMBL3822501)copy SMILEScopy InChI
Affinity DataIC50: 656nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183568(CHEMBL3823369)copy SMILEScopy InChI
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183567(CHEMBL3823177)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183573(CHEMBL3822843)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183517(CHEMBL3823859 | US11773085, Compound B50)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183454(CHEMBL3822539)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183451(CHEMBL3823551)copy SMILEScopy InChI
Affinity DataIC50: 2.98E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183452(CHEMBL3824351)copy SMILEScopy InChI
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of human BRD7 measured after mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183566(CHEMBL3822498)copy SMILEScopy InChI
Affinity DataIC50: 3.68E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183560(CHEMBL3822909)copy SMILEScopy InChI
Affinity DataIC50: 3.73E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183569(CHEMBL3823906)copy SMILEScopy InChI
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)copy SMILEScopy InChI
Affinity DataIC50: 3.85E+3nMAssay Description:Inhibition of TGFBR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183450(CHEMBL3824133)copy SMILEScopy InChI
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 5.09E+3nMAssay Description:Inhibition of ACVR1 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50157607(CHEMBL3753082 | US11773085, Compound B24)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human BRD9 isoform 1 co-expressed with H3 histone family 3A in HEK293 cells preincubated for 18 hrs followed by addition of nano-BRET f...More data for this Ligand-Target Pair
TargetActivin receptor type-1(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)copy SMILEScopy InChI
Affinity DataIC50: 5.13E+3nMAssay Description:Inhibition of ACVR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of TGFBR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 5.86E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 5.88E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50157607(CHEMBL3753082 | US11773085, Compound B24)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human BRD9 isoform 1 co-expressed with H4 histone in HEK293 cells preincubated for 18 hrs followed by addition of nano-BRET furimazine ...More data for this Ligand-Target Pair
TargetActivin receptor type-2B(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183449(CHEMBL3823101 | US11773085, Compound B23)copy SMILEScopy InChI
Affinity DataIC50: 7.68E+3nMAssay Description:Inhibition of ACVR2B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183566(CHEMBL3822498)copy SMILEScopy InChI
Affinity DataIC50: 9.34E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD2 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
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