Found 11 Enz. Inhib. hit(s) with all data for entry = 50047893 TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
3D Structure (crystal)TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 2.12E+3nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 2.18E+3nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 5.52E+3nMAssay Description:Competitive inhibition of post-glutamyl peptide hydrolyzing activity of human 20S proteasome using Cbz-Leu-Leu-Glu-AMC as substrate measured for 10 m...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 8.59E+3nMAssay Description:Competitive inhibition of post-glutamyl peptide hydrolyzing activity of human 20S proteasome using Cbz-Leu-Leu-Glu-AMC as substrate measured for 10 m...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 1.03E+4nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured for 10 mins by fluor...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 2.21E+4nMAssay Description:Competitive inhibition of trypsin-like activity of human 20S proteasome using Boc-Leu-Arg-Arg-AMC as substrate measured for 10 mins by fluorescence a...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataKi: 3.13E+4nMAssay Description:Competitive inhibition of post-glutamyl peptide hydrolyzing activity of human 20S proteasome using Cbz-Leu-Leu-Glu-AMC as substrate measured for 10 m...More data for this Ligand-Target Pair
