Compile Data Set for Download or QSAR
Found 40 Enz. Inhib. hit(s) with all data for entry = 50048126
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205397(CHEMBL3961192)copy SMILEScopy InChI
Affinity DataEC50:  270nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205562(CHEMBL3893457)copy SMILEScopy InChI
Affinity DataEC50:  3nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205445(CHEMBL3959152)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205469(CHEMBL3897216)copy SMILEScopy InChI
Affinity DataEC50:  0.480nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205470(CHEMBL3968025)copy SMILEScopy InChI
Affinity DataEC50:  6.5nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205471(CHEMBL3927718)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205473(CHEMBL3952126)copy SMILEScopy InChI
Affinity DataEC50:  0.140nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205474(CHEMBL3892208)copy SMILEScopy InChI
Affinity DataEC50:  0.430nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205476(CHEMBL3982830)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205478(CHEMBL3889524)copy SMILEScopy InChI
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205479(CHEMBL3925918)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205480(CHEMBL3936691)copy SMILEScopy InChI
Affinity DataEC50:  9nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205481(CHEMBL3952501)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205482(CHEMBL3943764)copy SMILEScopy InChI
Affinity DataEC50:  0.260nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205483(CHEMBL3935037)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205484(CHEMBL3901161)copy SMILEScopy InChI
Affinity DataEC50:  8.00E+4nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205485(CHEMBL3926685)copy SMILEScopy InChI
Affinity DataEC50:  9nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205486(CHEMBL3978552)copy SMILEScopy InChI
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205487(CHEMBL3947115)copy SMILEScopy InChI
Affinity DataEC50:  5nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205488(CHEMBL3917551)copy SMILEScopy InChI
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205489(CHEMBL3943114)copy SMILEScopy InChI
Affinity DataEC50:  1.80nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205490(CHEMBL3908747)copy SMILEScopy InChI
Affinity DataEC50:  40nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205491(CHEMBL3899701)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205492(CHEMBL3963609)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205493(CHEMBL3952665)copy SMILEScopy InChI
Affinity DataEC50:  0.180nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205494(CHEMBL3945422)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205495(CHEMBL3905849)copy SMILEScopy InChI
Affinity DataEC50:  1.80nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205496(CHEMBL3980962)copy SMILEScopy InChI
Affinity DataEC50:  0.600nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205497(CHEMBL3907204)copy SMILEScopy InChI
Affinity DataEC50:  0.700nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205498(CHEMBL3981277)copy SMILEScopy InChI
Affinity DataEC50:  0.650nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205499(CHEMBL3917072)copy SMILEScopy InChI
Affinity DataEC50:  400nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205500(CHEMBL3933984)copy SMILEScopy InChI
Affinity DataEC50:  0.130nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205501(CHEMBL3972297)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205502(CHEMBL3908085)copy SMILEScopy InChI
Affinity DataEC50:  18nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205503(CHEMBL3954145)copy SMILEScopy InChI
Affinity DataEC50:  7nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205558(CHEMBL3953544)copy SMILEScopy InChI
Affinity DataEC50:  0.600nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205559(CHEMBL3893937)copy SMILEScopy InChI
Affinity DataEC50:  200nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205560(CHEMBL3916470)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205561(CHEMBL3986815)copy SMILEScopy InChI
Affinity DataEC50:  500nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
UT Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50205410(CHEMBL3970245)copy SMILEScopy InChI
Affinity DataEC50:  0.0800nMAssay Description:Inhibition of porcupine-mediated Wnt signaling in mouse L-cells after 24 hrs by springerImage-Topflash reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KJRPubMed