Compile Data Set for Download or QSAR
Found 26 Enz. Inhib. hit(s) with all data for entry = 50048594
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224228(CHEMBL46233)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224175(CHEMBL48061)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224176(CHEMBL296963)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20321(3-[(4-tert-butylphenyl)methyl]-1-[(3-fluoro-4-meth...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224234(CHEMBL45252)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224229(CHEMBL48998)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224232(CHEMBL296729)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224196(CHEMBL43723)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224237(CHEMBL431341)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224230(CHEMBL47282)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224239(CHEMBL295773)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224100(CHEMBL44057)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224235(CHEMBL45417)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224226(CHEMBL45455)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224238(CHEMBL47602)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224195(CHEMBL48102)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224194(CHEMBL47473)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20284(CHEMBL391997 | CPZ | Capsazepine | N-[2-(4-chlorop...)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224193(CHEMBL295302)copy SMILEScopy InChI
Affinity DataIC50: 770nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224236(CHEMBL47241)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224099(CHEMBL45050)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224227(CHEMBL47820)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224231(CHEMBL48338)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50305278(CHEMBL595069 | iodoresiniferatoxin)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50224233(CHEMBL45817)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+4nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23B6294PubMed