Compile Data Set for Download or QSAR
Found 14 Enz. Inhib. hit(s) with all data for entry = 50048782
LigandPNGBDBM50227383(CHEMBL556758)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
LigandPNGBDBM50226939(CHEMBL36616)copy SMILEScopy InChI
Affinity DataKi:  0.240nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
LigandPNGBDBM50227384(CHEMBL172132)copy SMILEScopy InChI
Affinity DataKi:  0.420nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
LigandPNGBDBM50226938(CHEMBL38829)copy SMILEScopy InChI
Affinity DataKi:  0.690nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
LigandPNGBDBM50226961(CHEMBL38788)copy SMILEScopy InChI
Affinity DataKi:  0.960nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
LigandPNGBDBM50226937(CHEMBL289153)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50227384(CHEMBL172132)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
LigandPNGBDBM50226964(CHEMBL41064)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50226961(CHEMBL38788)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50226939(CHEMBL36616)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50226938(CHEMBL38829)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha-1 adrenergic receptor site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50226964(CHEMBL41064)copy SMILEScopy InChI
Affinity DataKi:  8.40nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50227383(CHEMBL556758)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha-1 adrenergic receptor site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt and Colman plc

Curated by ChEMBL
LigandPNGBDBM50226937(CHEMBL289153)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha-1 adrenergic receptor in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7QNKPubMed