TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]DAMGO from MOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3H]U69593 from KOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 168nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 313nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 602nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 793nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataEC50: 72nMAssay Description:Agonist activity at MOR (unknown origin) by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School of Pharmacy
Curated by ChEMBL
West Virginia University School of Pharmacy
Curated by ChEMBL
Affinity DataEC50: 253nMAssay Description:Agonist activity at MOR (unknown origin) by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair