Compile Data Set for Download or QSAR
Found 73 Enz. Inhib. hit(s) with all data for entry = 50049313
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238882(CHEMBL4094600)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238893(CHEMBL4096379)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human CLK4 expressed in baculovirus infected Sf21 cellsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50026622(CHEMBL408982)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238868(CHEMBL4072795)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238881(CHEMBL4067143)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238884(CHEMBL4060440)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238887(CHEMBL4093503)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human CLK2 (144 to 498 residues) expressed in insect cells using S6 kinase/Rsk2 substrate peptide 2 in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238892(CHEMBL4104765)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Compound was tested in vitro for its affinity towards rat striatal Dopamine receptor D2 labeled with [3H]- spiperoneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238883(CHEMBL4088668)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238885(CHEMBL4069124)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238886(CHEMBL4104122)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50026622(CHEMBL408982)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238893(CHEMBL4096379)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 138nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238866(CHEMBL4079878)copy SMILEScopy InChI
Affinity DataIC50: 139nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238892(CHEMBL4104765)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238879(CHEMBL4064426)copy SMILEScopy InChI
Affinity DataIC50: 155nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238880(CHEMBL4086890)copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238882(CHEMBL4094600)copy SMILEScopy InChI
Affinity DataIC50: 177nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238874(CHEMBL4100703)copy SMILEScopy InChI
Affinity DataIC50: 186nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238876(CHEMBL4081470)copy SMILEScopy InChI
Affinity DataIC50: 189nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238883(CHEMBL4088668)copy SMILEScopy InChI
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238881(CHEMBL4067143)copy SMILEScopy InChI
Affinity DataIC50: 245nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238868(CHEMBL4072795)copy SMILEScopy InChI
Affinity DataIC50: 257nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238888(CHEMBL4063617)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238886(CHEMBL4104122)copy SMILEScopy InChI
Affinity DataIC50: 283nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238885(CHEMBL4069124)copy SMILEScopy InChI
Affinity DataIC50: 404nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238866(CHEMBL4079878)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238890(CHEMBL4092984)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238875(CHEMBL4072220)copy SMILEScopy InChI
Affinity DataIC50: 439nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238889(CHEMBL4082710)copy SMILEScopy InChI
Affinity DataIC50: 529nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 690nMAssay Description:Inhibition of human DYRK1BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238870(CHEMBL4104093)copy SMILEScopy InChI
Affinity DataIC50: 993nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238876(CHEMBL4081470)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238884(CHEMBL4060440)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238887(CHEMBL4093503)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238880(CHEMBL4086890)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of recombinant human CDK9 expressed in fall armyworm sf21 cells using PDKtide as substrate in presence of [gamma-32]-ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of recombinant human GSK3beta expressed in fall armyworm sf21 cells using Phospho-glycogen synthase peptide-2 as substrate in presence of ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238879(CHEMBL4064426)copy SMILEScopy InChI
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238890(CHEMBL4092984)copy SMILEScopy InChI
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238888(CHEMBL4063617)copy SMILEScopy InChI
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238889(CHEMBL4082710)copy SMILEScopy InChI
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238878(CHEMBL4078073)copy SMILEScopy InChI
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 5.59E+3nMAssay Description:Opioid receptor affinity against Opioid receptor kappa 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238867(CHEMBL4083249)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DYRK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center for Biotherapy

Curated by ChEMBL
LigandPNGBDBM50238877(CHEMBL4059498)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1P55PubMed
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