Compile Data Set for Download or QSAR
Found 78 Enz. Inhib. hit(s) with all data for entry = 5482
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86616(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86614(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM31837(2,4-Bisanilinopyrimidine, 10 | Aurora Inhibitor, 3...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM50337135(4-((5,11-dimethyl-6-oxo-6,11-dihydro-5H-benzo[e]py...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86615(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86613(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM81552(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86601(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 7)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86602(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 8)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86598(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 3)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM50337135(4-((5,11-dimethyl-6-oxo-6,11-dihydro-5H-benzo[e]py...)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86599(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 4)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86606(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase C(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86610(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 10.7nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86622(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 11.6nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86611(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 11.9nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86623(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 13.4nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86614(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 14.3nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86615(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 14.5nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86609(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 14.9nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86601(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 7)copy SMILEScopy InChI
Affinity DataIC50: 15.2nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM50241089(2-(ethyl(3-(4-(5-(2-(3-fluorophenylamino)-2-oxoeth...)copy SMILEScopy InChI
Affinity DataIC50: 15.5nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86600(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 5)copy SMILEScopy InChI
Affinity DataIC50: 16.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86617(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 16.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase C(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)copy SMILEScopy InChI
Affinity DataIC50: 18.3nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86604(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 9)copy SMILEScopy InChI
Affinity DataIC50: 18.4nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM81552(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 18.4nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86602(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 8)copy SMILEScopy InChI
Affinity DataIC50: 18.7nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86610(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 19.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)copy SMILEScopy InChI
Affinity DataIC50: 19.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)copy SMILEScopy InChI
Affinity DataIC50: 23.2nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86616(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 24.2nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase C(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM81552(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 24.6nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase C(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM50241089(2-(ethyl(3-(4-(5-(2-(3-fluorophenylamino)-2-oxoeth...)copy SMILEScopy InChI
Affinity DataIC50: 25.3nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86598(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 3)copy SMILEScopy InChI
Affinity DataIC50: 25.9nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86599(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 4)copy SMILEScopy InChI
Affinity DataIC50: 28.6nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86609(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 36.7nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86604(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 9)copy SMILEScopy InChI
Affinity DataIC50: 39.3nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase C(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86598(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 3)copy SMILEScopy InChI
Affinity DataIC50: 40.5nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86613(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 43.7nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86600(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 5)copy SMILEScopy InChI
Affinity DataIC50: 45.1nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86608(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 53.2nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86611(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 55.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86618(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 2...)copy SMILEScopy InChI
Affinity DataIC50: 81.7nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86605(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 83.9nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase B(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86606(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 84.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Harvard Medical School

LigandPNGBDBM86607(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)copy SMILEScopy InChI
Affinity DataIC50: 86.8nMAssay Description:In vitro kinase assay of Aurora A, B, and C using Z-LYTE technology (Invitrogen) and ATP at Km apparent for each kinase.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6HZGPubMed
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