Compile Data Set for Download or QSAR
Found 29 Enz. Inhib. hit(s) with all data for entry = 6112
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109264(US8609710, 40)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109265(US8609710, 35 (2S,4R form))copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109258(US8609710, 34 (2S,4S form))copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109254(US8609710, 25)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109256(US8609710, 33)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109252(US8609710, 15 (2S form))copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109253(US8609710, 24)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109238(US8609710, 2)copy SMILEScopy InChI
Affinity DataIC50: 8.30nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109239(US8609710, 3)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109263(US8609710, 39)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109262(US8609710, 38)copy SMILEScopy InChI
Affinity DataIC50: 9.80nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109260(US8609710, 36)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109249(US8609710, 13)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109250(US8609710, 14)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109247(US8609710, 11)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109240(US8609710, 4)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109245(US8609710, 9)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109244(US8609710, 8)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109261(US8609710, 37)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109246(US8609710, 10)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109255(US8609710, 26)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109242(US8609710, 6)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109237(US8609710, 1)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109248(US8609710, 12)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109243(US8609710, 7)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109257(US8609710, 34 (2R,4S form))copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109241(US8609710, 5)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109251(US8609710, 15 (2R form))copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Daiichi Sankyo Company, Limited

US Patent
LigandPNGBDBM109259(US8609710, 35 (2R,4R form))copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Enzyme inhibition assay using TAFIa.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5DPPUS Patent