Compile Data Set for Download or QSAR
Found 39 Enz. Inhib. hit(s) with all data for entry = 6581
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139926(US8901087, 2)copy SMILEScopy InChI
Affinity DataKi:  0.0500nM ΔG°:  -58.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139933(US8901087, 27)copy SMILEScopy InChI
Affinity DataKi:  0.120nM ΔG°:  -56.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139959(US8901087, 191)copy SMILEScopy InChI
Affinity DataKi:  0.140nM ΔG°:  -56.2kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139951(US8901087, 95)copy SMILEScopy InChI
Affinity DataKi:  0.160nM ΔG°:  -55.9kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139952(US8901087, 97)copy SMILEScopy InChI
Affinity DataKi:  0.170nM ΔG°:  -55.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139925(US8901087, 1)copy SMILEScopy InChI
Affinity DataKi:  0.170nM ΔG°:  -55.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139946(US8901087, 76)copy SMILEScopy InChI
Affinity DataKi:  0.180nM ΔG°:  -55.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM46008(US8901087, 96)copy SMILEScopy InChI
Affinity DataKi:  0.190nM ΔG°:  -55.5kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139941(US8901087, 63)copy SMILEScopy InChI
Affinity DataKi:  0.220nM ΔG°:  -55.1kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139930(US8901087, 11)copy SMILEScopy InChI
Affinity DataKi:  0.300nM ΔG°:  -54.4kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139939(US8901087, 57)copy SMILEScopy InChI
Affinity DataKi:  0.330nM ΔG°:  -54.1kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139931(US8901087, 13)copy SMILEScopy InChI
Affinity DataKi:  0.400nM ΔG°:  -53.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139961(US8901087, 211)copy SMILEScopy InChI
Affinity DataKi:  0.440nM ΔG°:  -53.4kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139942(US8901087, 65)copy SMILEScopy InChI
Affinity DataKi:  0.450nM ΔG°:  -53.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139948(US8901087, 80)copy SMILEScopy InChI
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139950(US8901087, 91)copy SMILEScopy InChI
Affinity DataKi:  0.530nM ΔG°:  -52.9kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139929(US8901087, 8)copy SMILEScopy InChI
Affinity DataKi:  0.680nM ΔG°:  -52.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139938(US8901087, 53)copy SMILEScopy InChI
Affinity DataKi:  0.700nM ΔG°:  -52.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139932(US8901087, 25)copy SMILEScopy InChI
Affinity DataKi:  0.700nM ΔG°:  -52.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139958(US8901087, 181)copy SMILEScopy InChI
Affinity DataKi:  0.800nM ΔG°:  -51.9kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139956(US8901087, 141)copy SMILEScopy InChI
Affinity DataKi:  0.820nM ΔG°:  -51.9kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139927(US8901087, 3)copy SMILEScopy InChI
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139935(US8901087, 42)copy SMILEScopy InChI
Affinity DataKi:  1.03nM ΔG°:  -51.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139957(US8901087, 159)copy SMILEScopy InChI
Affinity DataKi:  1.25nM ΔG°:  -50.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139943(US8901087, 67)copy SMILEScopy InChI
Affinity DataKi:  1.25nM ΔG°:  -50.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139953(US8901087, 98)copy SMILEScopy InChI
Affinity DataKi:  1.43nM ΔG°:  -50.5kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139962(US8901087, 215)copy SMILEScopy InChI
Affinity DataKi:  1.80nM ΔG°:  -49.9kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139940(US8901087, 61)copy SMILEScopy InChI
Affinity DataKi:  2.46nM ΔG°:  -49.1kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139928(US8901087, 4)copy SMILEScopy InChI
Affinity DataKi:  3.10nM ΔG°:  -48.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139960(US8901087, 203)copy SMILEScopy InChI
Affinity DataKi:  3.16nM ΔG°:  -48.5kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139955(US8901087, 105)copy SMILEScopy InChI
Affinity DataKi:  3.40nM ΔG°:  -48.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139954(US8901087, 104)copy SMILEScopy InChI
Affinity DataKi:  3.63nM ΔG°:  -48.2kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139937(US8901087, 51)copy SMILEScopy InChI
Affinity DataKi:  5.10nM ΔG°:  -47.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139949(US8901087, 82)copy SMILEScopy InChI
Affinity DataKi:  5.84nM ΔG°:  -47.0kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139936(US8901087, 47)copy SMILEScopy InChI
Affinity DataKi:  6.40nM ΔG°:  -46.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139934(US8901087, 40)copy SMILEScopy InChI
Affinity DataKi:  7.95nM ΔG°:  -46.2kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139945(US8901087, 71)copy SMILEScopy InChI
Affinity DataKi:  9.12nM ΔG°:  -45.9kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139944(US8901087, 69)copy SMILEScopy InChI
Affinity DataKi:  9.36nM ΔG°:  -45.8kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme Corp.

US Patent
LigandPNGBDBM139947(US8901087, 77)copy SMILEScopy InChI
Affinity DataKi:  16.3nM ΔG°:  -44.5kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24B301WUS Patent