Compile Data Set for Download or QSAR
Found 46 Enz. Inhib. hit(s) with all data for entry = 7466
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196676(US9212171, 1)copy SMILEScopy InChI
Affinity DataEC50:  60nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196724(US9212171, 46)copy SMILEScopy InChI
Affinity DataEC50:  103nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196678(US9212171, 3)copy SMILEScopy InChI
Affinity DataEC50:  38nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196679(US9212171, 4)copy SMILEScopy InChI
Affinity DataEC50:  61nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196680(US9212171, 5)copy SMILEScopy InChI
Affinity DataEC50:  528nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196681(US9212171, 6)copy SMILEScopy InChI
Affinity DataEC50:  130nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196682(US9212171, 7)copy SMILEScopy InChI
Affinity DataEC50:  137nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196683(US9212171, 8)copy SMILEScopy InChI
Affinity DataEC50:  390nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196684(US9212171, 9)copy SMILEScopy InChI
Affinity DataEC50:  34nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196685(US9212171, 10)copy SMILEScopy InChI
Affinity DataEC50:  247nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196686(US9212171, 11)copy SMILEScopy InChI
Affinity DataEC50:  58nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196687(US9212171, 12)copy SMILEScopy InChI
Affinity DataEC50:  113nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196688(US9212171, 13)copy SMILEScopy InChI
Affinity DataEC50:  98nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196689(US9212171, 14)copy SMILEScopy InChI
Affinity DataEC50:  212nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196690(US9212171, 15)copy SMILEScopy InChI
Affinity DataEC50:  179nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196691(US9212171, 16)copy SMILEScopy InChI
Affinity DataEC50:  573nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196692(US9212171, 17)copy SMILEScopy InChI
Affinity DataEC50:  132nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196693(US9212171, 18)copy SMILEScopy InChI
Affinity DataEC50:  414nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196694(US9212171, 19)copy SMILEScopy InChI
Affinity DataEC50:  96nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196695(US9212171, 20)copy SMILEScopy InChI
Affinity DataEC50:  90nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196696(US9212171, 21)copy SMILEScopy InChI
Affinity DataEC50:  188nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196697(US9212171, 22)copy SMILEScopy InChI
Affinity DataEC50:  59nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196698(US9212171, 23)copy SMILEScopy InChI
Affinity DataEC50:  90nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196699(US9212171, 24)copy SMILEScopy InChI
Affinity DataEC50:  39nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196700(US9212171, 25)copy SMILEScopy InChI
Affinity DataEC50:  35nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196701(US9212171, 26)copy SMILEScopy InChI
Affinity DataEC50:  265nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196702(US9212171, 27)copy SMILEScopy InChI
Affinity DataEC50:  47nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196703(US9212171, 28)copy SMILEScopy InChI
Affinity DataEC50:  24nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196705(US9212171, 29)copy SMILEScopy InChI
Affinity DataEC50:  78nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196706(US9212171, 30 | US9212171, 32)copy SMILEScopy InChI
Affinity DataEC50:  33nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196707(US9212171, 31)copy SMILEScopy InChI
Affinity DataEC50:  25nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196706(US9212171, 30 | US9212171, 32)copy SMILEScopy InChI
Affinity DataEC50:  48nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196711(US9212171, 33)copy SMILEScopy InChI
Affinity DataEC50:  52nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196712(US9212171, 34 | US9212171, 36)copy SMILEScopy InChI
Affinity DataEC50:  185nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196713(US9212171, 35)copy SMILEScopy InChI
Affinity DataEC50:  101nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196712(US9212171, 34 | US9212171, 36)copy SMILEScopy InChI
Affinity DataEC50:  84nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196715(US9212171, 37)copy SMILEScopy InChI
Affinity DataEC50:  84nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196716(US9212171, 38 | US9212171, 40)copy SMILEScopy InChI
Affinity DataEC50:  69nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196717(US9212171, 39)copy SMILEScopy InChI
Affinity DataEC50:  141nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196716(US9212171, 38 | US9212171, 40)copy SMILEScopy InChI
Affinity DataEC50:  89nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196719(US9212171, 41)copy SMILEScopy InChI
Affinity DataEC50:  68nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196720(US9212171, 42)copy SMILEScopy InChI
Affinity DataEC50:  57nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196721(US9212171, 43)copy SMILEScopy InChI
Affinity DataEC50:  146nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196722(US9212171, 44)copy SMILEScopy InChI
Affinity DataEC50:  88nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196723(US9212171, 45)copy SMILEScopy InChI
Affinity DataEC50:  65nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Homo sapiens (Human))
HOFFMANN-LA ROCHE INC.

US Patent
LigandPNGBDBM196677(US9212171, 2)copy SMILEScopy InChI
Affinity DataEC50:  981nMT: 2°CAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25Q4TWHUS Patent